Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin

Aim: To compare ultrastructure, phenotypic profile and cell cycle progression ofMCF-7 human breast cancer cells and MCF7 sublines resistant to cisplatin (MCF-7/DDP) and doxorubicin (MCF-7/DOX). Methods: MTT-test, immunocytochemistry, flow cytometry, electron microscopy. Results: The development of...

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Veröffentlicht in:Experimental Oncology
Datum:2009
Hauptverfasser: Lukyanova, N.Yu., Rusetskya, N.V., Tregubova, N.A., Chekhun, V.F.
Format: Artikel
Sprache:English
Veröffentlicht: Інститут експериментальної патології, онкології і радіобіології ім. Р.Є. Кавецького НАН України 2009
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Online Zugang:https://nasplib.isofts.kiev.ua/handle/123456789/135701
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Назва журналу:Digital Library of Periodicals of National Academy of Sciences of Ukraine
Zitieren:Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin / N.Yu. Lukyanova, N.V. Rusetskya, N.A. Tregubova, V.F. Chekhun // Experimental Oncology. — 2009. — Т. 31, № 2. — С. 87–91. — Бібліогр.: 26 назв. — англ.

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Digital Library of Periodicals of National Academy of Sciences of Ukraine
id nasplib_isofts_kiev_ua-123456789-135701
record_format dspace
spelling Lukyanova, N.Yu.
Rusetskya, N.V.
Tregubova, N.A.
Chekhun, V.F.
2018-06-15T14:03:43Z
2018-06-15T14:03:43Z
2009
Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin / N.Yu. Lukyanova, N.V. Rusetskya, N.A. Tregubova, V.F. Chekhun // Experimental Oncology. — 2009. — Т. 31, № 2. — С. 87–91. — Бібліогр.: 26 назв. — англ.
1812-9269
https://nasplib.isofts.kiev.ua/handle/123456789/135701
Aim: To compare ultrastructure, phenotypic profile and cell cycle progression ofMCF-7 human breast cancer cells and MCF7 sublines resistant to cisplatin (MCF-7/DDP) and doxorubicin (MCF-7/DOX). Methods: MTT-test, immunocytochemistry, flow cytometry, electron microscopy. Results: The development of drug resistance to cisplatin and doxorubicin in MCF-7 cells upon the culturing of the initial cells with the raising concentrations of cytostatics was accompanied by the increase in cells adhesion, the increasing differentiation grade and the loss of steroid hormone receptors. Besides, it was shown that antiapoptotic mechanisms (decrease ofBcl-2 expression) and intracellular glutathione detoxifying system are involved in the process of cisplatin resistance development inMCF-7 cells. Atthe same time, P-glycoprotein overexpression in cells resistant to doxorubicin suggests MDR-dependent mechanism. Both doxorubicin- and cisplatin-resistant cells are characterized by the changes in the expression of several cell cycle regulators — Ki-67, cyclin D1, pRb and р21). Conclusion: The long-time culture of MCF-7 cells with cytostatic drugs results in the decreased cyclin D1, pRb, and Ki-67 expression and increased р21 expression with the increasing differentiation grade of the resistant cells. The underlying mechanisms of resistance to cisplatin and doxorubicin in MCF-7 cells may be different.
This work was supported by Fundamental researches state foundation (№ F28.4/047). We gratefully acknowledge Phd.M.P. Zavelevich (R.E. Kavetsky Institute of Experimental Pathology, Oncology and Radiobiology) for his helpful advice.
en
Інститут експериментальної патології, онкології і радіобіології ім. Р.Є. Кавецького НАН України
Experimental Oncology
Original contributions
Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
Article
published earlier
institution Digital Library of Periodicals of National Academy of Sciences of Ukraine
collection DSpace DC
title Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
spellingShingle Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
Lukyanova, N.Yu.
Rusetskya, N.V.
Tregubova, N.A.
Chekhun, V.F.
Original contributions
title_short Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
title_full Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
title_fullStr Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
title_full_unstemmed Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
title_sort molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin
author Lukyanova, N.Yu.
Rusetskya, N.V.
Tregubova, N.A.
Chekhun, V.F.
author_facet Lukyanova, N.Yu.
Rusetskya, N.V.
Tregubova, N.A.
Chekhun, V.F.
topic Original contributions
topic_facet Original contributions
publishDate 2009
language English
container_title Experimental Oncology
publisher Інститут експериментальної патології, онкології і радіобіології ім. Р.Є. Кавецького НАН України
format Article
description Aim: To compare ultrastructure, phenotypic profile and cell cycle progression ofMCF-7 human breast cancer cells and MCF7 sublines resistant to cisplatin (MCF-7/DDP) and doxorubicin (MCF-7/DOX). Methods: MTT-test, immunocytochemistry, flow cytometry, electron microscopy. Results: The development of drug resistance to cisplatin and doxorubicin in MCF-7 cells upon the culturing of the initial cells with the raising concentrations of cytostatics was accompanied by the increase in cells adhesion, the increasing differentiation grade and the loss of steroid hormone receptors. Besides, it was shown that antiapoptotic mechanisms (decrease ofBcl-2 expression) and intracellular glutathione detoxifying system are involved in the process of cisplatin resistance development inMCF-7 cells. Atthe same time, P-glycoprotein overexpression in cells resistant to doxorubicin suggests MDR-dependent mechanism. Both doxorubicin- and cisplatin-resistant cells are characterized by the changes in the expression of several cell cycle regulators — Ki-67, cyclin D1, pRb and р21). Conclusion: The long-time culture of MCF-7 cells with cytostatic drugs results in the decreased cyclin D1, pRb, and Ki-67 expression and increased р21 expression with the increasing differentiation grade of the resistant cells. The underlying mechanisms of resistance to cisplatin and doxorubicin in MCF-7 cells may be different.
issn 1812-9269
url https://nasplib.isofts.kiev.ua/handle/123456789/135701
citation_txt Molecular profile and cell cycle in mcf-7 cells resistant to cisplatin and doxorubicin / N.Yu. Lukyanova, N.V. Rusetskya, N.A. Tregubova, V.F. Chekhun // Experimental Oncology. — 2009. — Т. 31, № 2. — С. 87–91. — Бібліогр.: 26 назв. — англ.
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