Hit identification of FGFR1 inhibitors using receptor-based virtual screening
Aim. To identify novel FGFR1 inhibitors using the virtual screening approach. Methods. Virtual screening of a small organic compounds library was performed by molecular docking using the Autodock 4.2.6 program package. The compounds activity was determined by in vitro biochemical tests using γ-32P A...
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| Published in: | Вiopolymers and Cell |
|---|---|
| Date: | 2019 |
| Main Authors: | Tarnavskiy, S.S., Protopopov, M.V., Borovykov, O.V., Pryhodko, A.O., Bdzhola, V.G., Yarmoluk, S.M. |
| Format: | Article |
| Language: | English |
| Published: |
Інститут молекулярної біології і генетики НАН України
2019
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| Subjects: | |
| Online Access: | https://nasplib.isofts.kiev.ua/handle/123456789/154388 |
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| Journal Title: | Digital Library of Periodicals of National Academy of Sciences of Ukraine |
| Cite this: | Hit identification of FGFR1 inhibitors using receptor-based virtual screening / S.S. Tarnavskiy, M.V. Protopopov, O.V. Borovykov, A.O. Pryhodko, V.G. Bdzhola, S.M. Yarmoluk // Вiopolymers and Cell. — 2019. — Т. 35, № 2. — С. 143-151. — Бібліогр.: 24 назв. — англ. |
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