Донори Н2S у створенні інноваційних лікарських засобів

Fundamental studies have identified a new group of gaseous signaling molecules – the so-called gasotransmitters – NO, CO, and H2S, which are involved in the regulation of a large number of metabolic processes. The results of these studies allowed determining a new direction in medicinal/pharmaceutic...

Full description

Saved in:
Bibliographic Details
Date:2017
Main Authors: Kaminskyy, D. V., Kryshchyshyn, A. P., Yelisyeyeva, O. P., Lesyk, R. B.
Format: Article
Language:Ukrainian
Published: National University of Pharmacy 2017
Subjects:
Online Access:https://ophcj.nuph.edu.ua/article/view/ophcj.17.918
Tags: Add Tag
No Tags, Be the first to tag this record!
Journal Title:Journal of Organic and Pharmaceutical Chemistry

Institution

Journal of Organic and Pharmaceutical Chemistry
Description
Summary:Fundamental studies have identified a new group of gaseous signaling molecules – the so-called gasotransmitters – NO, CO, and H2S, which are involved in the regulation of a large number of metabolic processes. The results of these studies allowed determining a new direction in medicinal/pharmaceutical chemistry – creation of hydrogen sulfide donor compounds as potential drugs. The article presents the main achievements in the search for new H2S donors: the main stages of H2S metabolism and its biological effects; the classes of compounds that can release hydrogen sulfide based on the nature of sulfur-containing functional groups as well as the mechanism of H2S releasing. Additionally, the characteristic of the most successful direction – creation of the so-called hybrid molecules is given. The latter are compounds bearing fragments of the well known drugs covalently bounded with groups being capable to release H2S.