Оптимізація та масштабування методу синтезу похідних азаіндолу

In this study, an optimized method for the synthesis of azaindoles was developed and successfully scaled up to a 100 g batch. Improved yields were observed when using electron-deficient azaheterocycles and substrates bearing electron-withdrawing substituents. 6-Chloro-1H-pyrrolo[3,2-c]pyridine was s...

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Datum:2025
Hauptverfasser: Kordubailo, Mykyta V., Tolmachev, Andrey A.
Format: Artikel
Sprache:English
Veröffentlicht: National University of Pharmacy 2025
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Online Zugang:https://ophcj.nuph.edu.ua/article/view/323307
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Назва журналу:Journal of Organic and Pharmaceutical Chemistry

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Journal of Organic and Pharmaceutical Chemistry